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Table 1 List of drug formulated in Tablet-in-Tablet or compressed-coated tablet

From: Review on Tablet in Tablet techniques

Active ingredient

Category/use

Excipients

References

Paliperidone

Antipsychotic

HPC-H, Euragit RL-PO, Glycerylbehenate, MCC, HPMC-K100 M

[15]

Orlistat and venlafaxine

Antiobesity and antidepressant

For core tablet—βCD, SD Mannitol, Ludiflash, Kollidon CLF, Kollidon-30, SLS, Sucrose, Talc, Mg-Stearate, Cherry Flavour, Methyl Paraben

For outer coating—βCD, Eudragit EPO, Ludipress LCE, Maltodextrin, Xanthan Gum, Kollidon-30,Citric Acid,Sucralose, Peppermint flavor, Propyl Paraben, Talc, Mg.Sterate

[9]

Amoxicillin and potassium clavulanate

Antibacterial and β lactamase inhibitors

Steric acid and avicel layer

[17]

Acetaminophen

Analgesic and antipyretic

HPMC, Mg.Sterate, Lactose-crystal cellulose

[11]

Glipizide

Antidiabetic

βCD, HPC-L, HPC-M, MCC, Eudragit RL PO, Mg.Sterate

[5]

Nifedipine

Antihypertensive, calcium channel blockers

HPC-L, HPC-M, Eudragit RSPO, Mg.Sterate

[6]

Prednisolone

Immuno-suppressant

Carboxymethyl xanthan gum, Sodium alginate, Calcium chloride, MCC,Polyplasdone XL, Tri-Sodium Citrate, Trisodium orthophosphate dodecahydrate, Mg.Sterate.

[8].

Carvedilol

Antihypertensive or non-selective beta adrenergic receptor blocker

Polyoxy Ethylene Oxide WSR 205, HPMC K4M, MCC, Sodium starch glycollate, Mg.Sterate.

[14]