Compounds | BBB | CYP2D6 substrate | CYP3A4 substrate | CYP1A2 inhibitor | AMES toxicity | Oral Toxicity (LD50) | Hepatotoxicity | Skin Sensitization |
---|---|---|---|---|---|---|---|---|
Artelinic acid |  − 0.70 | No | No | Yes | No | 2.44 | No | No |
Artemiside | 0.07 | No | Yes | Yes | No | 2.55 | Yes | No |
Artemisone | 0.30 | No | Yes | No | No | 2.89 | Yes | No |
Artemotil | 1.38 | No | Yes | No | No | 3.19 | Yes | No |
Artenimol | 0.26 | No | Yes | No | Yes | 2.52 | No | No |
Caffeic acid | 0.88 | No | Yes | Yes | No | 2.51 | No | No |
Caftaric acid | 0.89 | no | No | yes | no | 2.46 | No | No |
Chicoric acid | 0.54 | No | Yes | Yes | No | 2.10 | No | No |
Chlorogenic acid | 0.97 | No | No | Yes | No | 2.44 | No | No |
Echinacoside | 0.71 | No | Yes | Yes | No | 2.55 | Yes | No |